I-BET151

• Supplier: Creative Biomart
• Catalog: EI-0410
• Cas Number: 1300031-49-5
• Formula: C 23 H 21 N 5 O 3
• Molecular Weight: 434.27
• Purity: ≥95% by HPLC
• Description: A BET bromodomain inhibitor that interacts with BRD4 and BRD3 BET proteins and displaces them from chromatin; displays high efficacy against human and murine MLL-fusion leukemic cell lines, through the induction of early cell cycle arrest and apoptosis