PDGFR/VEGFR2 Tyrosine Kinase Inhibitor, 5-Br SU6668 - CAS 251356-32-8 - Calbiochem
| Name | PDGFR/VEGFR2 Tyrosine Kinase Inhibitor, 5-Br SU6668 - CAS 251356-32-8 - Calbiochem |
|---|---|
| Supplier | EMD Millipore |
| Catalog | 521236 |
| Cas Number | 251356-32-8 |
| Formula | C₁₈H₁₇BrN₂O₃ |
| Purity | ≥97% by HPLC |
| Description | A cell-permeable, ATP-binding pocket-targeting, 5-bromoindolinone analog of SU6668 (Cat. No. 521235) that is equally potent as SU6668 in inhibiting PDGFR (IC 50 = 60 nM against PDGFRβ), while exhibiting more enhanced activity against VEGFR2 and FGFR1 (IC 50 = 1.73 and 2.05 µM, respectively) in cell-free kinase assays |
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