RXRα Inhibitor, K-80003 - Calbiochem

Name RXRα Inhibitor, K-80003 - Calbiochem
Supplier EMD Millipore
Catalog 557451
Formula C₂₃H₂₃FO₂
Purity ≥95% by HPLC
Description A cell permeable, Sulindac analog with IC 50 =2.4 µM for RXRα binding, and unlike other NSAIDs, is inactive toward COX2 and COX1 even at 1 mM. The compound displays potent inhibition of RXRα dependent AKT Activation in both PC3 and A549 cells, and is RXRα but not RXRγ expression dependent as shown in PC3 cells
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