HMTase Inhibitor IV, UNC0638 - Calbiochem
| Name | HMTase Inhibitor IV, UNC0638 - Calbiochem |
|---|---|
| Supplier | EMD Millipore |
| Catalog | 382192 |
| Formula | C₃₀H₄₇N₅O₂ |
| Purity | ≥99% by HPLC |
| Description | A cell-permeable quinazolinamine compound that acts as a potent and reversible inhibitor of G9a and GLP HMTases (histone methyltransferases) (IC 50 = ≤ 15 and 19 nM for G9a and GLP, respectively) and displays ~15-fold greater selectivity over DNMT1 and minimally blocks the activities of JMJD2E (IC 50 = 4.66 µM) and SETD7, SETD8, PRMT3 and SUV39H2 (IC 50 > 10 µM) |
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