BRD2 Inhibitor II, BIC1 - Calbiochem

• Supplier: EMD Millipore
• Catalog: 203830
• Formula: C₁₇H₁₆N₄S₂
• Purity: ≥95% by HPLC
• Description: A cell-permeable benzimidazolyl-benzimidazolothione that targets BD1 (bromodomain 1) of the BET (bromodomain and extra terminal domain) family member BRD2 ( K d = 28 µM in equilibrium binding studies by SPR, using human BRD2 aa 74-194), making it inaccessible for acetylated H4K12 (histone H4 Lys12) binding

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