PIM-Kinase Inhibitor X, CX-6258 - Calbiochem

• Supplier: EMD Millipore
• Catalog: 526529
• Formula: C₂₆H₂₄ClN₃O₃•HCl
• Purity: ≥99% by HPLC
• Description: An orally bioavailable oxindolo-furanyl compound that acts as a potent, reversible and ATP-competitive inhibitor of pan PIM-kinases (IC 50 = 5, 25 and 16 nM for PIM-1, PIM-2 and PIM-3, respectively; K i = 5 nM for PIM-1) with excellent selectivity over 107 kinases (IC 80 > 500 nM)

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