BD 1047 dihydrobromide

• Supplier: R&D Systems
• Catalog: 0956
• Prices: $129.00, $535.00
• Sizes: 10 mg, 50 mg
• Cas Number: 138356-21-5
• Chemical Name: N-[2-(3,4-Dichlorophenyl)ethyl]-N-methyl-2-(dimethylamino)ethylaminedihydrobromide
• Formula: C13H20Cl2N2.2HBr
• Molecular Weight: 437.04
• Purity: >99%

Product References

The ON:OFF switch, sigma1R-HINT1 protein, controls GPCR-NMDA receptor - The ON:OFF switch, sigma1R-HINT1 protein, controls GPCR-NMDA receptor

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Effects of BD1047, a sigma1 receptor antagonist, on the expression of mTOR, - Effects of BD1047, a sigma1 receptor antagonist, on the expression of mTOR,

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Sigma-1 receptor antagonism restores injury-induced decrease of voltage-gated - Sigma-1 receptor antagonism restores injury-induced decrease of voltage-gated

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NOP receptor mediates anti-analgesia induced by agonist-antagonist opioids. - NOP receptor mediates anti-analgesia induced by agonist-antagonist opioids.

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The calcium-sensitive Sigma-1 receptor prevents cannabinoids from provoking - The calcium-sensitive Sigma-1 receptor prevents cannabinoids from provoking

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Dynamic interaction between sigma-1 receptor and Kv1.2 shapes neuronal and - Dynamic interaction between sigma-1 receptor and Kv1.2 shapes neuronal and

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Decreases in cocaine self-administration with dual inhibition of the dopamine - Decreases in cocaine self-administration with dual inhibition of the dopamine

Hiranita T, Soto PL, Kohut SJ, Kopajtic T, Cao J, Newman AH, Tanda G, Katz JL. J Pharmacol Exp Ther. 2011 Nov;339(2):662-77.

Sigma-1 Receptor Antagonist BD1047 Reduces Allodynia and Spinal ERK - Sigma-1 Receptor Antagonist BD1047 Reduces Allodynia and Spinal ERK

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Intrathecal injection of the neurosteroid, DHEAS, produces mechanical allodynia - Intrathecal injection of the neurosteroid, DHEAS, produces mechanical allodynia

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