JTV 519 fumarate

• Supplier: R&D Systems
• Catalog: 4564
• Prices: $155.00, $645.00
• Sizes: 10 mg, 50 mg
• Chemical Name: 1-(2,3-Dihydro-7-methoxy-1,4-benzothiazepin-4(5H)-yl)-3-[4-(phenylmethyl)-1-piperidinyl]-1-propanonefumarate
• Formula: C25H32N2O2.C4H4O4
• Molecular Weight: 540.67
• Purity: >98%

Product References

K201 (JTV519) suppresses spontaneous Ca2+ release and [3H]ryanodine binding to - K201 (JTV519) suppresses spontaneous Ca2+ release and [3H]ryanodine binding to

Hunt DJ, Jones PP, Wang R, Chen W, Bolstad J, Chen K, Shimoni Y, Chen SR. Biochem J. 2007 Jun 15;404(3):431-8.

Effect of K201, a novel antiarrhythmic drug on calcium handling and - Effect of K201, a novel antiarrhythmic drug on calcium handling and

Chen YJ, Chen YC, Wongcharoen W, Lin CI, Chen SA. Br J Pharmacol. 2008 Mar;153(5):915-25. Epub 2007 Nov 12.

Designing calcium release channel inhibitors with enhanced electron donor - Designing calcium release channel inhibitors with enhanced electron donor

Ye Y, Yaeger D, Owen LJ, Escobedo JO, Wang J, Singer JD, Strongin RM, Abramson JJ. Mol Pharmacol. 2012 Jan;81(1):53-62.