G-1

Name	G-1
Supplier	R&D Systems
Catalog	3577
Prices	$189.00, $765.00
Sizes	10 mg, 50 mg
Cas Number	881639-98-1
Chemical Name	(±)-1-[(3aR,4S,9bS*)-4-(6-Bromo-1,3-benzodioxol-5-yl)-3a,4,5,9b-tetrahydro-3H-cyclopenta[c]quinolin-8-yl]-ethanone
Formula	C21H18BrNO3
Molecular Weight	412.28
Purity	>98%
Supplier Page	Shop

Product References

A calixpyrrole derivative acts as an antagonist to GPER, a G-protein coupled - A calixpyrrole derivative acts as an antagonist to GPER, a G-protein coupled

Lappano R, Rosano C, Pisano A, Santolla MF, De Francesco EM, De Marco P, Dolce V, Ponassi M, Felli L, Cafeo G, Kohnke FH, Abonante S, Maggiolini M. Dis Model Mech. 2015 Oct 1;8(10):1237-46.

SIRT1 is involved in oncogenic signaling mediated by GPER in breast cancer. - SIRT1 is involved in oncogenic signaling mediated by GPER in breast cancer.

Santolla MF, Avino S, Pellegrino M, De Francesco EM, De Marco P, Lappano R, Vivacqua A, Cirillo F, Rigiracciolo DC, Scarpelli A, Abonante S, Maggiolini M. Cell Death Dis. 2015 Jul 30;6:e1834.

GPER agonist G-1 decreases adrenocortical carcinoma (ACC) cell growth in vitro - GPER agonist G-1 decreases adrenocortical carcinoma (ACC) cell growth in vitro

Chimento A, Sirianni R, Casaburi I, Zolea F, Rizza P, Avena P, Malivindi R, De Luca A, Campana C, Martire E, Domanico F, Fallo F, Carpinelli G, Cerquetti L, Amendola D, Stigliano A, Pezzi V. Oncotarget. 2015 Aug 7;6(22):19190-203.

Estrogen accelerates the resolution of inflammation in macrophagic cells. - Estrogen accelerates the resolution of inflammation in macrophagic cells.

Villa A, Rizzi N, Vegeto E, Ciana P, Maggi A. Sci Rep. 2015 Oct 19;5:15224.

Acquisition of epithelial-mesenchymal transition phenotype in the - Acquisition of epithelial-mesenchymal transition phenotype in the

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GPR30 activation decreases anxiety in the open field test but not in the elevated - GPR30 activation decreases anxiety in the open field test but not in the elevated

Anchan D, Clark S, Pollard K, Vasudevan N. Brain Behav. 2014 Jan;4(1):51-9.

Activation of a Gq-coupled membrane estrogen receptor rapidly attenuates - Activation of a Gq-coupled membrane estrogen receptor rapidly attenuates

Nag S, Mokha SS. Neuroscience. 2014 May 16;267:122-34.

Estrogen rapidly enhances incisional pain of ovariectomized rats primarily - Estrogen rapidly enhances incisional pain of ovariectomized rats primarily

An G, Li W, Yan T, Li S. Int J Mol Sci. 2014 Jun 11;15(6):10479-91.

Selective GPER activation decreases proliferation and activates apoptosis in - Selective GPER activation decreases proliferation and activates apoptosis in

Chimento A, Casaburi I, Bartucci M, Patrizii M, Dattilo R, Avena P, Ando S, Pezzi V, Sirianni R. Cell Death Dis. 2013 Aug 1;4:e747.

Seven transmembrane G protein-coupled receptor repertoire of gastric ghrelin - Seven transmembrane G protein-coupled receptor repertoire of gastric ghrelin

Engelstoft MS, Park WM, Sakata I, Kristensen LV, Husted AS, Osborne-Lawrence S, Piper PK, Walker AK, Pedersen MH, Nohr MK, Pan J, Sinz CJ, Carrington PE, Akiyama TE, Jones RM, Tang C, Ahmed K, Offermanns S, Egerod KL, Zigman JM, Schwartz TW. Mol Metab. 2013 Sep 4;2(4):376-92.