| Name | A 887826 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 4571 |
| Prices | $189.00, $765.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Blocker |
| Cas Number | 1266212-81-0 |
| Chemical Name | 5-(4-Butoxy-3-chlorophenyl)-N-[[2-(4-morpholinyl)-3-pyridinyl]methyl-3-pyridinecarboxamide |
| Formula | C26H29ClN4O3 |
| Molecular Weight | 480.99 |
| Purity | >97 % |
| Description | Potent voltage-dependent Na V 1.8 channel blocker (IC 50 = 11 nM in recombinant human Na V 1.8 channels). Reduces tactile allodynia in neuropathic rat models. 3- and 28-fold more potent at Na V 1.8 channels compared to Na V 1.2 and Na V 1.7 channels respectively. |
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