| Name | ABP 688 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 1297 |
| Prices | $149.00, $629.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 924298-51-1 |
| Chemical Name | 3-[2-(6-Methyl-2-pyridinyl)ethynyl]-2-cyclohexene-1-oneO-methyloxime |
| Formula | C15H16N2O |
| Molecular Weight | 240.3 |
| Purity | >98 % |
| Description | High affinity human mGlu 5 receptor antagonist (K i = 1.7 nM). Inhibits glutamate-induced calcium release from L(tk-) cells expressing human mGlu 5 receptors (IC 50 = 2.3 nM). |
| Supplier Page | Shop |
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Orozco LD, Liu H, Perkins E, Johnson DA, Chen BB, Fan F, Baker RC, Roman RJ. J Pharmacol Exp Ther. 2013 Jul;346(1):67-74.