AdTx1

Name AdTx1
Supplier Tocris Bioscience
Catalog 5096
Prices $205.00
Sizes 10 µg
Function Type Antagonist
Formula C310H481N87O100S8
Molecular Weight 7283.22
Description Selective, high affinity, non-competitive α 1A adrenoceptor antagonist (K i = 0.35 nM). Exhibits no significant activity against a range of other GPCRs, including α 2A , β 1 and β 2 adrenoceptors . Antagonizes effects of phenylephrine (Cat. No. 2838) on isolated rabbit prostate muscle in vitro and on intra-urethral pressure in rats.
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Product References

Structural basis of a potent peptide inhibitor designed for Kv1.3 channel, a - Structural basis of a potent peptide inhibitor designed for Kv1.3 channel, a

Han S, Yi H, Yin SJ, Chen ZY, Liu H, Cao ZJ, Wu YL, Li WX. J Biol Chem. 2008 Jul 4;283(27):19058-65.

Selective inhibition of CCR7(-) effector memory T cell activation by a novel - Selective inhibition of CCR7(-) effector memory T cell activation by a novel

Li Z, Liu WH, Han S, Peng BW, Yin J, Wu YL, He XH, Li WX. J Biol Chem. 2012 Aug 24;287(35):29479-94.