Name | Amlodipine besylate |
---|---|
Supplier | Tocris Bioscience |
Catalog | 4857 |
Prices | $95.00 |
Sizes | 50 mg |
Function Type | Blocker |
Cas Number | 111470-99-6 |
Chemical Name | 2-[(2-Aminoethoxy)methyl]-4-(2-chlorophenyl)-1,4-dihydro-6-methyl-3,5-pyridinedicarboxylicacid3-ethyl5-methylesterbenzenesulfonate |
Formula | C20H25ClN2O5.C6H6O3S |
Molecular Weight | 567.05 |
Purity | >99 % |
Description | L-type calcium channel blocker that displays antihypertensive properties. Inhibits Ca 2+ -induced contractions in depolarized rat aorta (IC 50 = 1.9 nM) and displays vasoprotective effects in cardiovascular disease. Inhibits proliferation of human vascular smooth muscle cells and epidermoid carcinoma A431 cells (IC 50 = 25 μ M). |
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