Amthamine dihydrobromide

• Supplier: Tocris Bioscience
• Catalog: 3989
• Prices: $139.00, $585.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 142457-00-9
• Chemical Name: 2-Amino-5-(2-aminoethyl)-4-methylthiazoledihydrobromide
• Formula: C6H11N3S.2HBr
• Molecular Weight: 319.06
• Purity: >99 %
• Description: Highly selective H 2 agonist, slightly more potent than histamine itself. Only a weak antagonist at H 3 and has no activity at H 1 receptors. Induces vasodilation of cerebral arteries and decreases myogenic tone in vitro .

Product References

Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative - Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative

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The new potent and selective histamine H2 receptor agonist amthamine as a tool to - The new potent and selective histamine H2 receptor agonist amthamine as a tool to

Coruzzi G, Timmerman H, Adami M, Bertaccini G. Naunyn Schmiedebergs Arch Pharmacol. 1993 Jul;348(1):77-81.

In vitro cardiac pharmacology of the new histamine H2-receptor agonist amthamine: - In vitro cardiac pharmacology of the new histamine H2-receptor agonist amthamine:

Poli E, Pozzoli C, Coruzzi G, Bertaccini G, Timmerman H. Agents Actions. 1993 Sep;40(1-2):44-9.

Histamine decreases myogenic tone in rat cerebral arteries by - Histamine decreases myogenic tone in rat cerebral arteries by

Jarajapu YP, Oomen C, Uteshev VV, Knot HJ. Eur J Pharmacol. 2006 Oct 10;547(1-3):116-24. Epub 2006 Jul 27.