Apamin

Name Apamin
Supplier Tocris Bioscience
Catalog 0104
Prices $289.00
Sizes 1 mg
Function Type Inhibitor
Cas Number 24345-16-2
Formula C79H131N31O24S4
Molecular Weight 2027.34
Description Prototypical potent and highly selective inhibitor of the small-conductance Ca 2+ -activated K + -channel (K Ca 2, SK). Blocks medium after-hyperpolarization in vitro and is brain penetrant and convulsive in vivo .
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Product References

Apamin. - Apamin.

Habermann E. Pharmacol Ther. 1984;25(2):255-70.

Potassium channel toxins. - Potassium channel toxins.

Strong PN. Pharmacol Ther. 1990;46(1):137-62.

Behavioral effects of apamin, a selective inhibitor of the SK(Ca)-channel, in - Behavioral effects of apamin, a selective inhibitor of the SK(Ca)-channel, in

van der Staay FJ, Fanelli RJ, Blokland A, Schmidt BH. Neurosci Biobehav Rev. 1999 Dec;23(8):1087-110.

Matching molecules to function: neuronal Ca2+-activated K+ channels and - Matching molecules to function: neuronal Ca2+-activated K+ channels and

Stocker M, Hirzel K, D'hoedt D, Pedarzani P. Toxicon. 2004 Jun 15;43(8):933-49.