Name | AR-C 102222 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 1445 |
Prices | $225.00, $925.00 |
Sizes | 10 mg, 50 mg |
Function Type | Inhibitor |
Cas Number | 253771-21-0 |
Chemical Name | 5-[(4'-Amino-5',8'-difluorospiro[piperidine-4,2'(1'H)-quinaxolin]-1-yl)carbonyl]-2-pyridinecarbonitrilehydrochloride |
Formula | C19H16F2N6O.HCl |
Molecular Weight | 418.83 |
Purity | >98 % |
Description | Inducible nitric oxide synthase (iNOS) inhibitor; selective for iNOS over eNOS (IC 50 values are 0.037 and >100 μ M for iNOS and eNOS respectively). Exhibits antinociceptive and anti-inflammatory activity in rodent pain models. |
Supplier Page | Shop |
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