Arvanil

• Supplier: Tocris Bioscience
• Catalog: 2668
• Prices: $69.00, $245.00
• Sizes: 5 mg, 25 mg
• Function Type: Agonist
• Cas Number: 128007-31-8
• Chemical Name: N-[(4-Hydroxy-3-methoxyphenyl)methyl]-5Z,8Z,11Z,14Z-eicosatetraenamide
• Formula: C28H41NO3
• Molecular Weight: 439.64
• Purity: >98 %
• Description: Cannabinoid CB 1 and vanilloid TRPV1 (VR1) agonist (K i values are 0.5 and 0.3 μ M respectively). Also inhibits the anandamide transporter (IC 50 = 3.6 μ M). Analgesic, vasodilatory and anti-inflammatory in vivo .

Product References

Unsaturated long-chain N-acyl-vanillyl-amides (N-AVAMs): vanilloid receptor - Unsaturated long-chain N-acyl-vanillyl-amides (N-AVAMs): vanilloid receptor

Melck D, Bisogno T, De Petrocellis L, Chuang H, Julius D, Bifulco M, Di Marzo V. Biochem Biophys Res Commun. 1999 Aug 19;262(1):275-84.

Neurobehavioral activity in mice of N-vanillyl-arachidonyl-amide. - Neurobehavioral activity in mice of N-vanillyl-arachidonyl-amide.

Di Marzo V, Breivogel C, Bisogno T, Melck D, Patrick G, Tao Q, Szallasi A, Razdan RK, Martin BR. Eur J Pharmacol. 2000 Oct 20;406(3):363-74.

New perspectives on enigmatic vanilloid receptors. - New perspectives on enigmatic vanilloid receptors.

Szallasi A, Di Marzo V. Trends Neurosci. 2000 Oct;23(10):491-7.