Name | ASP 7663 |
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Supplier | Tocris Bioscience |
Catalog | 5310 |
Prices | $185.00, $755.00 |
Sizes | 10 mg, 50 mg |
Function Type | Activator |
Cas Number | 1190217-35-6 |
Chemical Name | (2E)-2-[7-Fluoro-1,2-dihydro-1-(2-methylpropyl)-2-oxo-3H-indol-3-ylidene]aceticacid |
Formula | C14H14FNO3 |
Molecular Weight | 263.26 |
Purity | >98 % |
Description | Selective TRPA1 activator (EC 50 values are ~0.5 μ M in human, mouse and rat). Displays little or no affinity at more than 60 other related receptors, channels and enzymes. Stimulates 5-HT release from QGP-1 cells. Exhibits an abdominal analgesic effect in vivo . Orally bioavailable. |
Supplier Page | Shop |