AZD 9272

• Supplier: Tocris Bioscience
• Catalog: 5199
• Prices: $149.00, $629.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 327056-26-8
• Chemical Name: 3-Fluoro-5-[3-(5-fluoro-2-pyridinyl)-1,2,4-oxadiazol-5-yl]benzonitrile
• Formula: C14H6F2N4O
• Molecular Weight: 284.22
• Purity: >98 %
• Description: Potent and selective mGlu 5 antagonist (IC 50 values are 2.6 and 7.6 nM for rat and human receptors, respectively). Exhibits >3900-fold selectivity for mGlu 5 over other mGlu receptors. Also selective over a panel of other targets. Displays discriminative effects in rats. Orally bioavailable and brain penetrant.

Product References

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Azidothymidine is effective against human multiple myeloma: a new use for an old - Azidothymidine is effective against human multiple myeloma: a new use for an old

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