BA 1

Name BA 1
Supplier Tocris Bioscience
Catalog 2855
Prices $199.00
Sizes 1 mg
Function Type Agonist
Cas Number 183241-31-8
Formula C57H76N14O11
Molecular Weight 1133.32
Description Potent bombesin receptor subtype 3 (BRS-3; BB 3 ) agonist (IC 50 = 2.52 nM). Also GRPR (BB 1 ) and NMBR (BB 2 ) agonist (IC 50 values are 0.26 and 1.55 nM respectively). Enhances glucose transport in obese and diabetic primary myocytes. Also stimulates NCI-H1299 lung cancer cell proliferation in vitro .
Supplier Page Shop

Product References

Comparative pharmacology of bombesin receptor subtype-3, nonpeptide agonist - Comparative pharmacology of bombesin receptor subtype-3, nonpeptide agonist

Moreno P, Mantey SA, Nuche-Berenguer B, Reitman ML, Gonzalez N, Coy DH, Jensen RT. J Pharmacol Exp Ther. 2013 Oct;347(1):100-16.

Effect of bombesin receptor subtype-3 and its synthetic agonist on signaling, - Effect of bombesin receptor subtype-3 and its synthetic agonist on signaling,

Gonzalez N, Martin-Duce A, Martinez-Arrieta F, Moreno-Villegas Z, Portal-Nunez S, Sanz R, Egido J. Int J Mol Med. 2015 Apr;35(4):925-31.

ML-18 is a non-peptide bombesin receptor subtype-3 antagonist which inhibits lung - ML-18 is a non-peptide bombesin receptor subtype-3 antagonist which inhibits lung

Moody TW, Mantey SA, Moreno P, Nakamura T, Lacivita E, Leopoldo M, Jensen RT. Peptides. 2015 Feb;64:55-61.