| Name | BAZ2-ICR |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 3138 |
| Prices | $205.00, $845.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Chemical Name | 4-[4-(1-Methyl-1H-pyrazole-4-yl)-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-5-yl]benzonitrile |
| Formula | C20H19N7 |
| Molecular Weight | 357.41 |
| Purity | >98 % |
| Description | Selective BAZ2 bromodomain inhibitor (IC 50 values are 130 and 180 nM for BAZ2A and BAZ2B respectively). Exhibits 15-fold selectivity for the BAZ2 bromodomain over the CERC2 bromodomain and >100-fold selectivity over a range of other bromodomains. Accelerates FRAP recovery in a BAZ2A FRAP assay. |
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