BD 1008 dihydrobromide

Name BD 1008 dihydrobromide
Supplier Tocris Bioscience
Catalog 3875
Prices $139.00, $585.00
Sizes 10 mg, 50 mg
Cas Number 138356-09-9
Chemical Name N-[2-(3,4-Dichlorophenyl)ethyl]-N-methyl-2-(1-pyrrolidinyl)ethylaminedihydrobromide
Formula C15H22Cl2N2.2HBr
Molecular Weight 463.08
Description Potent and selective σ -ligand (K i against [ 3 H]-(+)-3-PPP = 0.34 nM).
Supplier Page Shop

Product References

Synthesis, characterization, and biological evaluation of a novel class of - Synthesis, characterization, and biological evaluation of a novel class of

de Costa BR, Radesca L, Di Paolo L, Bowen WD. J Med Chem. 1992 Jan;35(1):38-47.

Differentiation of sigma ligand-activated receptor subtypes that modulate - Differentiation of sigma ligand-activated receptor subtypes that modulate

Monnet FP, de Costa BR, Bowen WD. Br J Pharmacol. 1996 Sep;119(1):65-72.

Antagonism of N-methyl-D-aspartate receptors by sigma site ligands: potency, - Antagonism of N-methyl-D-aspartate receptors by sigma site ligands: potency,

Whittemore ER, Ilyin VI, Woodward RM. J Pharmacol Exp Ther. 1997 Jul;282(1):326-38.