nor -Binaltorphimine dihydrochloride

• Supplier: Tocris Bioscience
• Catalog: 4048
• Prices: $159.00, $665.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 113158-34-2
• Chemical Name: 17,17'-(Dicyclopropylmethyl)-6,6',7,7'-6,6'-imino-7,7'-binorphinan-3,4',14,14'-tetroldihydrochloride
• Formula: C40H43N3O6.2HCl
• Molecular Weight: 734.72
• Purity: >98 %
• Description: A selective κ -opioid receptor antagonist.

Product References

Structure-activity relationship of N17'-substituted norbinaltorphimine congeners. - Structure-activity relationship of N17'-substituted norbinaltorphimine congeners.

Portoghese PS, Lin CE, Farouz-Grant F, Takemori AE. J Med Chem. 1994 May 13;37(10):1495-500.

Differential agonist regulation of the human kappa-opioid receptor. - Differential agonist regulation of the human kappa-opioid receptor.

Blake AD, Bot G, Li S, Freeman JC, Reisine T. J Neurochem. 1997 May;68(5):1846-52.

Nor-binaltorphimine precipitates withdrawal and excitatory amino acid release in - Nor-binaltorphimine precipitates withdrawal and excitatory amino acid release in

Feng Y, Rockhold RW, Ho IK. J Pharmacol Exp Ther. 1997 Nov;283(2):932-8.