BQ-3020

Name BQ-3020
Supplier Tocris Bioscience
Catalog 1188
Prices $219.00
Sizes 500 µg
Function Type Agonist
Cas Number 143113-45-5
Formula C96H140N20O25S
Molecular Weight 2006.35
Description Highly potent and selective ET B endothelin receptor agonist (K i values are 0.18 and 970 nM at human ET B and ET A receptors respectively).
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Product References

Distinct subdomains of human endothelin receptors determine their selectivity to - Distinct subdomains of human endothelin receptors determine their selectivity to

Sakamoto A, Yanagisawa M, Sawamura T, Enoki T, Ohtani T, Sakurai T, Nakao K, Toyo-oka T, Masaki T. J Biol Chem. 1993 Apr 25;268(12):8547-53.

Effects of selective ETB-receptor stimulation on arterial, venous and capillary - Effects of selective ETB-receptor stimulation on arterial, venous and capillary

Ekelund U, Adner M, Edvinsson L, Mellander S. Br J Pharmacol. 1994 Jul;112(3):887-94.

[3H]BQ-123, a highly specific and reversible radioligand for the endothelin ETA - [3H]BQ-123, a highly specific and reversible radioligand for the endothelin ETA

Ihara M, Yamanaka R, Ohwaki K, Ozaki S, Fukami T, Ishikawa K, Towers P, Yano M. Eur J Pharmacol. 1995 Feb 14;274(1-3):1-6.

Pharmacological differences between rat and human endothelin B receptors. - Pharmacological differences between rat and human endothelin B receptors.

Reynolds EE, Hwang O, Flynn MA, Welch KM, Cody WL, Steinbaugh B, He JX, Chung FZ, Doherty AM. Biochem Biophys Res Commun. 1995 Apr 17;209(2):506-12.