| Name | 3-Bromocytisine |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 0427 |
| Prices | $199.00, $825.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Agonist |
| Cas Number | 207390-14-5 |
| Chemical Name | (1R,5S)-9-Bromo-1,2,3,4,5,6-hexahydro-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one |
| Formula | C11H13BrN2O |
| Molecular Weight | 269.14 |
| Purity | >98 % |
| Description | Potent agonist of α 4 β 4, α 4 β 2 and α 7 nACh receptors (IC 50 values are 0.28, 0.30 and 31.6 nM respectively). Displays different effects on high (HS) and low (LS) ACh sensitivity α 4 β 2 nAChRs (EC 50 values are 0.008 and 0.05 μ M respectively). |
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Houlihan LM, Slater Y, Guerra DL, Peng JH, Kuo YP, Lukas RJ, Cassels BK, Bermudez I. J Neurochem. 2001 Sep;78(5):1029-43.
Moroni M, Zwart R, Sher E, Cassels BK, Bermudez I. Mol Pharmacol. 2006 Aug;70(2):755-68. Epub 2006 May 23.