Name | Cantharidin |
---|---|
Supplier | Tocris Bioscience |
Catalog | 3281 |
Prices | $129.00 |
Sizes | 50 mg |
Function Type | Inhibitor |
Cas Number | 56-25-7 |
Chemical Name | (3aα,4β,7β,7aα)-Hexahydro-3a,7a-dimethyl-4,7-epoxyisobenzofuran-1,3-dione |
Formula | C10H12O4 |
Molecular Weight | 196.2 |
Description | Natural toxin inhibitor of protein phosphatases 1 and 2A (K i values are 1.1 and 0.19 μ M respectively); similar to okadaic acid (Cat. No. 1136). Displays > 500-fold selectivity over PP2B. |
Supplier Page | Shop |
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Knapp J, Boknik P, Luss I, Huke S, Linck B, Luss H, Muller FU, Muller T, Nacke P, Noll T, Piper HM, Schmitz W, Vahlensieck U, Neumann J. J Pharmacol Exp Ther. 1999 Jun;289(3):1480-6.