Name | Capsazepine |
---|---|
Supplier | Tocris Bioscience |
Catalog | 0462 |
Prices | $159.00, $665.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 138977-28-3 |
Chemical Name | N-[2-(4-Chlorophenyl)ethyl]-1,3,4,5-tetrahydro-7,8-dihydroxy-2H-2-benzazepine-2-carbothioamide |
Formula | C19H21ClN2O2S |
Molecular Weight | 376.9 |
Purity | >99 % |
Description | Selective vanilloid receptor antagonist (K i = 3.2 μ M). Inhibits carrageenan inflammation-induced hyperalgesic responses in the rat. Also activates amiloride-sensitive epithelial Na + channel ENaC δ . Also available as part of the Vanilloid TRPV1 Receptor Tocriset™ . |
Supplier Page | Shop |
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