| Name | CCF 642 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 0452 |
| Prices | $125.00, $525.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 346640-08-2 |
| Chemical Name | 3-(4-Methoxyphenyl)-5-[(5-nitro-2-thienyl)methylene]-2-thioxo-4-thiazolidinone |
| Formula | C15H10N2O4S3 |
| Molecular Weight | 378.45 |
| Purity | >98 % |
| Description | Protein disulfide isomerase (PDI) inhibitor. Induces acute ER stress and apoptosis in multiple myeloma cells in vitro (submicromolar activity). Prolongs survival of C57BL/KaLwRij mice engrafted with 5TGM1-luc myeloma. Also a bone marrow-sparing compound. |
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