CGP 39551

• Supplier: Tocris Bioscience
• Catalog: 1469
• Prices: $169.00, $705.00
• Sizes: 10 mg, 50 mg
• Function Type: Antagonist
• Cas Number: 127910-32-1
• Chemical Name: (E)-(±)-2-Amino-4-methyl-5-phosphono-3-pentenoicacidethylester
• Formula: C8H16NO5P
• Molecular Weight: 237.19
• Purity: >98 %
• Description: Potent, selective and competitive NMDA antagonist (K i = 310 nM for inhibition of [ 3 H]-CPP binding in rat brain). Centrally active upon oral administration in vivo .

Product References

CGP 37849 and CGP 39551: novel and potent competitive N-methyl-D-aspartate - CGP 37849 and CGP 39551: novel and potent competitive N-methyl-D-aspartate

Fagg GE, Olpe HR, Pozza MF, Baud J, Steinmann M, Schmutz M, Portet C, Baumann P, Thedinga K, Bittiger H, et al.. Br J Pharmacol. 1990 Apr;99(4):791-7.

Anticonvulsant and behavioral effects of two novel competitive - Anticonvulsant and behavioral effects of two novel competitive

Loscher W, Honack D. J Pharmacol Exp Ther. 1991 Feb;256(2):432-40.

Effects of competitive NMDA receptor antagonists on excitatory amino acid-evoked - Effects of competitive NMDA receptor antagonists on excitatory amino acid-evoked

D'Hooge R, Raes A, Van de Vijver G, Van Bogaert PP, De Deyn PP. Fundam Clin Pharmacol. 1999;13(1):67-74.