CGP 74514 dihydrochloride

• Supplier: Tocris Bioscience
• Catalog: 2199
• Prices: $155.00, $645.00
• Sizes: 10 mg, 50 mg
• Function Type: Inhibitor
• Chemical Name: rel-N2-[(1R,2S)-2-Aminocyclohexyl]-N6-(3-chlorophenyl)-9-ethyl-9H-purine-2,6-diaminedihydrochloride
• Formula: C19H24ClN7.2HCl
• Molecular Weight: 458.82
• Purity: >98 %
• Description: Potent cdk1 inhibitor (IC 50 = 25 nM). Reduces Akt phosphorylation and increases mitochondrial damage in leukemia cells in vitro in combination with LY 294002 .

Product References

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Synthesis, radiolabelling and biological characterization of - Synthesis, radiolabelling and biological characterization of

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