Name | CGS 12066B dimaleate |
---|---|
Supplier | Tocris Bioscience |
Catalog | 1169 |
Prices | $89.00, $375.00 |
Sizes | 10 mg, 50 mg |
Function Type | Agonist |
Cas Number | 109028-10-6 |
Chemical Name | 7-Trifluoromethyl-4-(4-methyl-1-piperazinyl)pyrrolo[1,2-a]-quinoxalinedimaleate |
Formula | C17H17F3N4.2C4H4O4 |
Molecular Weight | 566.49 |
Purity | >98 % |
Description | 5-HT 1B full agonist, 10-fold selective over 5-HT 1A and 1000-fold selective over 5-HT 2C receptors. Centrally active following systemic administration. |
Supplier Page | Shop |
Neale RF, Fallon SL, Boyar WC, Wasley JW, Martin LL, Stone GA, Glaeser BS, Sinton CM, Williams M. Eur J Pharmacol. 1987 Apr 7;136(1):1-9.
Schoeffter P, Hoyer D. Naunyn Schmiedebergs Arch Pharmacol. 1989 Jun;339(6):675-83.
Tomkins DM, O'Neill MF. Pharmacol Biochem Behav. 2000 May;66(1):129-36.