Name | CGS 15943 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 0638 |
Prices | $75.00, $255.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 104615-18-1 |
Chemical Name | 9-Chloro-2-(2-furanyl)-[1,2,4]triazolo[1,5-c]quinazolin-5-amine |
Formula | C13H8ClN5O |
Molecular Weight | 285.69 |
Purity | >99 % |
Description | Potent adenosine receptor antagonist (K i values are 3.5, 4.2, 16 and 51 nM for human A 1 , A 2A , A 2B and A 3 receptors respectively). Orally active in vivo . |
Supplier Page | Shop |
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Klotz KN. Naunyn Schmiedebergs Arch Pharmacol. 2000 Nov;362(4-5):382-91.