2-Chloro-N 6 -cyclopentyladenosine

Name 2-Chloro-N 6 -cyclopentyladenosine
Supplier Tocris Bioscience
Catalog 0443
Prices $139.00, $579.00
Sizes 10 mg, 50 mg
Function Type Agonist
Cas Number 37739-05-2
Chemical Name 2-Chloro-N-cyclopentyladenosine
Formula C15H20ClN5O4
Molecular Weight 369.81
Purity >98 %
Description Potent and selective adenosine A 1 receptor agonist (K i values are 0.8, 2300 and 42 nM for human A 1 , A 2A and A 3 receptors respectively; EC 50 = 18800 nM for hA 2B ). Centrally active following systemic administration in vivo .
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Product References

2-Chloro-N6-cyclopentyladenosine: a highly selective agonist at A1 adenosine - 2-Chloro-N6-cyclopentyladenosine: a highly selective agonist at A1 adenosine

Lohse MJ, Klotz KN, Schwabe U, Cristalli G, Vittori S, Grifantini M. Naunyn Schmiedebergs Arch Pharmacol. 1988 Jun;337(6):687-9.

Anticonvulsant doses of 2-chloro-N6-cyclopentyladenosine, an adenosine A1 - Anticonvulsant doses of 2-chloro-N6-cyclopentyladenosine, an adenosine A1

Concas A, Santoro G, Mascia MP, Maciocco E, Dazzi L, Ongini E, Biggio G. J Pharmacol Exp Ther. 1993 Nov;267(2):844-51.

Pharmacology of the highly selective A1 adenosine receptor agonist - Pharmacology of the highly selective A1 adenosine receptor agonist

Monopoli A, Conti A, Dionisotti S, Casati C, Camaioni E, Cristalli G, Ongini E. Arzneimittelforschung. 1994 Dec;44(12):1305-12.

Adenosine receptors and their ligands. - Adenosine receptors and their ligands.

Klotz KN. Naunyn Schmiedebergs Arch Pharmacol. 2000 Nov;362(4-5):382-91.