Ciglitazone

Name Ciglitazone
Supplier Tocris Bioscience
Catalog 3327
Prices $189.00, $765.00
Sizes 10 mg, 50 mg
Function Type Agonist
Cas Number 74772-77-3
Chemical Name 5-[[4-[(1-Methylcyclohexyl)methoxy]phenyl]methyl]-2,4-thiazolidinedione
Formula C18H23NO3S
Molecular Weight 333.44
Purity >99 %
Description Selective agonist at PPAR γ (peroxisome proliferator-activated receptor γ ). Activates PPAR γ with an EC 50 value of 3 μ M in vitro , and is at least 33-fold selective over PPAR α and δ . Antihyperglycemic in vivo .
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Product References

The structure-activity relationship between peroxisome proliferator-activated - The structure-activity relationship between peroxisome proliferator-activated

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Thiazolidinediones--the new insulin enhancers. - Thiazolidinediones--the new insulin enhancers.

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Peroxisome proliferator-activated receptor gamma ligands are potent inhibitors of - Peroxisome proliferator-activated receptor gamma ligands are potent inhibitors of

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