Name | CINPA 1 |
---|---|
Supplier | Tocris Bioscience |
Catalog | 4119 |
Prices | $109.00, $459.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 102636-74-8 |
Chemical Name | Ethyl[5-[(diethylamino)acetyl]-10,11-dihydro-5H-dibenz[b,f]azepin-3-yl]carbamate |
Formula | C23H29N3O3 |
Molecular Weight | 395.49 |
Purity | >98 % |
Description | Potent CAR antagonist (IC 50 = 70 nM). Exhibits >90-fold selectivity for CAR over pregnane X receptor (PXR). Also selective over a panel of other nuclear receptors including FXR, LXR, PPAR γ and RXR. |
Supplier Page | Shop |