| Name | CMPD101 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 2186 |
| Prices | $139.00 |
| Sizes | 10 mg |
| Function Type | Inhibitor |
| Cas Number | 865608-11-3 |
| Chemical Name | 3-[[[4-Methyl-5-(4-pyridinyl)-4H-1,2,4-triazol-3-yl]methyl]amino]-N-[[2-(trifluoromethyl)phenyl]methyl]benzamide |
| Formula | C24H21F3N6O |
| Molecular Weight | 466.46 |
| Purity | >98 % |
| Description | Potent and selective GRK2/3 inhibitor (IC 50 values are 32 and 54 nM for GRK3 and GRK2, respectively). Exhibits selectivity for GRK2/3 over GRK1/5. Reduces DAMGO -induced desensitization and internalization of μ -opioid receptors. |
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