Name | α -Conotoxin MII |
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Supplier | Tocris Bioscience |
Catalog | 3119 |
Prices | $535.00 |
Sizes | 500 µg |
Function Type | Antagonist |
Cas Number | 175735-93-0 |
Formula | C67H103N23O22S4 |
Molecular Weight | 1710.99 |
Description | Highly potent and selective competitive antagonist for α 3 β 2 subunit-containing nicotinic receptors (IC 50 = 0.5 - 3.5 nM at α 3 β 2 expressed in Xenopus oocytes). Also potently blocks β 3-containing neuronal nicotinic receptors. Displays > 200-fold selectivity for α 3 β 2 over α 2 β 2, α 4 β 2 and α 3 β 4. |
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