| Name | CP 945598 hydrochloride |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 1317 |
| Prices | $225.00, $925.00 |
| Sizes | 10 mg, 50 mg |
| Function Type | Antagonist |
| Cas Number | 686347-12-6 |
| Chemical Name | 1-[8-(2-Chlorophenyl)-9-(4-chlorophenyl)-9H-purin-6-yl]-4-(ethylamino)piperidine-4-carboxamidehydrochloride |
| Formula | C25H25Cl2N7O.HCl |
| Molecular Weight | 546.88 |
| Purity | >99 % |
| Description | Selective, high affinity CB 1 antagonist (K i values are 0.7 and 0.12 nM in binding and functional assays respectively). Displays low affinity for CB 2 receptors (K i = 7600 nM). |
| Supplier Page | Shop |
Griffith DA, Hadcock JR, Black SC, Iredale PA, Carpino PA, DaSilva-Jardine P, Day R, DiBrino J, Dow RL, Landis MS, O'Connor RE, Scott DO. J Med Chem. 2009 Jan 22;52(2):234-7.
Hadcock JR, Griffith DA, Iredale PA, Carpino PA, Dow RL, Black SC, O'Connor R, Gautreau D, Lizano JS, Ward K, Hargrove DM, Kelly-Sullivan D, Scott DO. Biochem Biophys Res Commun. 2010 Apr 2;394(2):366-71. doi: