8-CPT-2Me-cAMP, sodium salt

Name 8-CPT-2Me-cAMP, sodium salt
Supplier Tocris Bioscience
Catalog 2688
Prices $175.00
Sizes 1 mg
Function Type Activator
Cas Number 634207-53-7
Chemical Name 8-(4-Chlorophenylthio)-2'-O-methyladenosine-3',5'-cyclicmonophosphatesodiumsalt
Formula C17H16ClN5O6PS.Na
Molecular Weight 507.82
Purity >99 %
Description Selective activator of Epac, the cAMP-sensitive guanine nucleotide-exchange factor for Rap1 and Rap2. Activates Epac1 (EC 50 = 2.2 μ M), but not PKA (EC 50 > 10 μ M). Stimulates Epac-mediated Ca 2+ -mediated Ca 2+ release in pancreatic β -cells in vitro . Cell permeable analog (Cat. No. 4853) also available.
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