CTAP

Name CTAP
Supplier Tocris Bioscience
Catalog 4726
Prices $149.00
Sizes 1 mg
Function Type Antagonist
Cas Number 103429-32-9
Formula C51H69N13O11S2
Molecular Weight 1104.32
Description Potent and selective μ opioid receptor antagonist (IC 50 = 3.5 nM). Displays > 1200-fold selectivity over δ opioid and somatostatin receptors. Brain penetrant and active in vivo .
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Product References

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Blood-brain barrier permeability and bioavailability of a highly potent and - Blood-brain barrier permeability and bioavailability of a highly potent and

Abbruscato TJ, Thomas SA, Hruby VJ, Davis TP. J Pharmacol Exp Ther. 1997 Jan;280(1):402-9.