Cyproheptadine hydrochloride

Name Cyproheptadine hydrochloride
Supplier Tocris Bioscience
Catalog 2601
Prices $95.00
Sizes 50 mg
Function Type Antagonist
Cas Number 969-33-5
Chemical Name 4-(5H-Dibenzo[a,d]cyclohepten-5-ylidine)-methylpiperidinehydrochloride
Formula C21H21N.HCl
Molecular Weight 323.86
Purity >98 %
Description Non-selective 5HT 2 antagonist, migraine prophylactic. Also SETD7/9 inhibitor (IC 50 = 1 μ M). Decreases expression and increases degradation of estrogen receptor (ER) α in breast tumor MCF7 cells. Inhibits growth of MCF7 xenografts in mice.
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Product References

International Union of Pharmacology classification of receptors for - International Union of Pharmacology classification of receptors for

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Inhibitory 5-hydroxytryptamine receptors involved in pressor effects obtained by - Inhibitory 5-hydroxytryptamine receptors involved in pressor effects obtained by

Moran A, Velasco C, Salvador T, Martin ML, San Roman L. Br J Pharmacol. 1994 Dec;113(4):1358-62.