(-)-Cytisine

• Supplier: Tocris Bioscience
• Catalog: 4520
• Prices: $89.00, $355.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 485-35-8
• Chemical Name: (1R,5S)-1,2,3,4,5,6-hexahydro-1,5-methano-8H-pyrido[1,2-a][1,5]diazocin-8-one
• Formula: C11H14N2O
• Molecular Weight: 190.24
• Purity: >99 %
• Description: A potent, selective agonist at neuronal nicotinic receptors. Acts as a partial agonist at β 2-containing nicotinic receptors.

Product References

Behavioural and pharmacokinetic studies on nicotine, cytisine and lobeline. - Behavioural and pharmacokinetic studies on nicotine, cytisine and lobeline.

Reavill C, Walther B, Stolerman IP, Testa B. Neuropharmacology. 1990 Jul;29(7):619-24.

Localization of nicotinic cholinergic receptors in rat brain: autoradiographic - Localization of nicotinic cholinergic receptors in rat brain: autoradiographic

Happe HK, Peters JL, Bergman DA, Murrin LC. Neuroscience. 1994 Oct;62(3):929-44.

Partial agonist properties of cytisine on neuronal nicotinic receptors containing - Partial agonist properties of cytisine on neuronal nicotinic receptors containing

Papke RL, Heinemann SF. Mol Pharmacol. 1994 Jan;45(1):142-9.