Deltorphin I

• Supplier: Tocris Bioscience
• Catalog: 5424
• Prices: $95.00
• Sizes: 1 mg
• Function Type: Agonist
• Cas Number: 122752-15-2
• Formula: C37H52N8O10
• Molecular Weight: 768.87
• Description: Potent δ -opioid receptor agonist (IC 50 = 0.5 nM in human granulocytes). Exhibits a high rate of blood-brain barrier penetrance.

Product References

Deltorphins: a family of naturally occurring peptides with high affinity and - Deltorphins: a family of naturally occurring peptides with high affinity and

Erspamer V, Melchiorri P, Falconieri-Erspamer G, Negri L, Corsi R, Severini C, Barra D, Simmaco M, Kreil G. Proc Natl Acad Sci U S A. 1989 Jul;86(13):5188-92.

[D-Ala2]deltorphin I binding and pharmacological evidence for a special subtype - [D-Ala2]deltorphin I binding and pharmacological evidence for a special subtype

Stefano GB, Melchiorri P, Negri L, Hughes TK Jr, Scharrer B. Proc Natl Acad Sci U S A. 1992 Oct 1;89(19):9316-20.

Deltorphin transport across the blood-brain barrier. - Deltorphin transport across the blood-brain barrier.

Fiori A, Cardelli P, Negri L, Savi MR, Strom R, Erspamer V. Proc Natl Acad Sci U S A. 1997 Aug 19;94(17):9469-74.