Diprenorphine

Name Diprenorphine
Supplier Tocris Bioscience
Catalog 0794
Prices $175.00
Sizes 50 mg
Function Type Antagonist
Cas Number 14357-78-9
Chemical Name 17-(Cyclopropylmethyl)-4,5-epoxy-18,19-dihydro-3-hydroxy-6-methoxy-α,α-dimethyl-6,14-ethenomorphinan-7-methanol
Formula C26H35NO4
Molecular Weight 425.56
Purity >99 %
Description Non-selective opioid receptor antagonist (K i values are 0.017, 0.072 and 0.23 nM for κ -, μ - and δ -opioid receptors).
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Product References

Classification of opioid receptors. - Classification of opioid receptors.

Paterson SJ, Robson LE, Kosterlitz HW. Br Med Bull. 1983 Jan;39(1):31-6.

The effect of the nonselective opioid antagonist diprenorphine on vasopressin - The effect of the nonselective opioid antagonist diprenorphine on vasopressin

Iwasaki Y, Gaskill MB, Boss CA, Robertson GL. Endocrinology. 1994 Jan;134(1):48-54.

Pharmacological characterization of the cloned kappa-, delta-, and mu-opioid - Pharmacological characterization of the cloned kappa-, delta-, and mu-opioid

Raynor K, Kong H, Chen Y, Yasuda K, Yu L, Bell GI, Reisine T. Mol Pharmacol. 1994 Feb;45(2):330-4.