Name | DQP 1105 |
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Supplier | Tocris Bioscience |
Catalog | 2168 |
Prices | $175.00, $709.00 |
Sizes | 10 mg, 50 mg |
Function Type | Antagonist |
Cas Number | 380560-89-4 |
Chemical Name | 5-(4-Bromophenyl)-3-(1,2-dihydro-6-methyl-2-oxo-4-phenyl-3-quinolinyl)-4,5-dihydro-γ-oxo-1H-pyrazole-1-butanoicacid |
Formula | C29H24BrN3O4 |
Molecular Weight | 558.42 |
Purity | >97 % |
Description | Noncompetitive NMDA receptor antagonist; displays over 50-fold selectivity for GluN2D- and GluN2C-containing receptors over GluN2B-, GluK2-, GluA1- and GluN2A-containing receptors (IC 50 values are 2.7, 8.5, 121, 153, 198 and 206 μ M, respectively). Reduces frequency of channel opening. |
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