| Name | DR 2313 |
|---|---|
| Supplier | Tocris Bioscience |
| Catalog | 4491 |
| Prices | $69.00, $149.00, $629.00 |
| Sizes | 1 mg, 10 mg, 50 mg |
| Function Type | Inhibitor |
| Cas Number | 284028-90-6 |
| Chemical Name | 1,5,7,8-Tetrahydro-2-methyl-4H-thiopyrano[4,3-d]pyrimidin-4-one |
| Formula | C8H10N2OS |
| Molecular Weight | 182.24 |
| Purity | >99 % |
| Description | Competitive inhibitor of poly(ADP-ribose) polymerase (PARP) (IC 50 values are 0.20 and 0.24 μ M for PARP-1 and PARP-2 respectively). Neuroprotective; reduces neuronal cell death in models of cerebral ischemia in vivo and in vitro . Brain penetrant. |
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