EHT 1864

Name EHT 1864
Supplier Tocris Bioscience
Catalog 1261
Prices $209.00, $879.00
Sizes 10 mg, 50 mg
Function Type Inhibitor
Cas Number 754240-09-0
Chemical Name 5-(5-(7-(Trifluoromethyl)quinolin-4-ylthio)pentyloxy)-2-(morpholinomethyl)-4H-pyran-4-onedihydrochloride
Formula C25H27F3N2O4S.2HCl
Molecular Weight 581.47
Purity >98 %
Description Inhibitor of Rac family GTPases. Blocks activation by direct binding to Rac1, Rac1b, Rac2 and Rac3 (K D values are 40, 50, 60 and 250 nM respectively). Inhibits Rac, Ras and Tiam-induced growth transformation of NIH-3T3 fibroblasts. Reduces β -amyloid peptide production in vivo .
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