Endomorphin-1

• Supplier: Tocris Bioscience
• Catalog: 3576
• Prices: $115.00
• Sizes: 5 mg
• Cas Number: 189388-22-5
• Formula: C34H38N6O5
• Molecular Weight: 610.67
• Description: Endogenous peptide with an exceptionally high affinity (K i = 360 pM) and selectivity for μ opioid receptors (4000- and 15000-fold preference over δ and κ respectively).

Product References

A potent and selective endogenous agonist for the mu-opiate receptor. - A potent and selective endogenous agonist for the mu-opiate receptor.

Zadina JE, Hackler L, Ge LJ, Kastin AJ. Nature. 1997 Apr 3;386(6624):499-502.

Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse - Pharmacological characterization of endomorphin-1 and endomorphin-2 in mouse

Goldberg IE, Rossi GC, Letchworth SR, Mathis JP, Ryan-Moro J, Leventhal L, Su W, Emmel D, Bolan EA, Pasternak GW. J Pharmacol Exp Ther. 1998 Aug;286(2):1007-13.

Differential effects of endomorphin-1, endomorphin-2, and Tyr-W-MIF-1 on - Differential effects of endomorphin-1, endomorphin-2, and Tyr-W-MIF-1 on

Harrison LM, Kastin AJ, Zadina JE. Peptides. 1998;19(4):749-53.

Parallel stimulations of in vitro and in situ [35S]GTPgammaS binding by - Parallel stimulations of in vitro and in situ [35S]GTPgammaS binding by

Kakizawa K, Shimohira I, Sakurada S, Fujimura T, Murayama K, Ueda H. Peptides. 1998;19(4):755-8.