Fentanyl citrate

• Supplier: Tocris Bioscience
• Catalog: 5525
• Prices: $69.00, $255.00
• Sizes: 10 mg, 50 mg
• Function Type: Agonist
• Cas Number: 990-73-8
• Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamidecitrate
• Formula: C22H28N2O.C6H8O7
• Molecular Weight: 528.59
• Purity: >99 %
• Description: Potent and selective μ -opioid receptor agonist (K i values are 7.0, 151 and 470 nM for μ -, δ - and κ -opioid receptors respectively). Displays antinociceptive activity in vivo .

Product References

Receptor reserve and affinity of mu opioid agonists in mouse antinociception: - Receptor reserve and affinity of mu opioid agonists in mouse antinociception:

Zernig G, Issaevitch T, Broadbear JH, Burke TF, Lewis JW, Brine GA, Woods JH. Life Sci. 1995;57(23):2113-25.

Opioid activity of C8813, a novel and potent opioid analgesic. - Opioid activity of C8813, a novel and potent opioid analgesic.

Liu ZH, Jin WQ, Dai QY, Chen XJ, Zhang HP, Chi ZQ. Life Sci. 2003 May 30;73(2):233-41.

Opioid interactions in rhesus monkeys: effects of delta + mu and delta + kappa - Opioid interactions in rhesus monkeys: effects of delta + mu and delta + kappa

Stevenson GW, Folk JE, Linsenmayer DC, Rice KC, Negus SS. J Pharmacol Exp Ther. 2003 Dec;307(3):1054-64. Epub 2003 Oct 13.