[D-Lys 3 ]-GHRP-6

Name [D-Lys 3 ]-GHRP-6
Supplier Tocris Bioscience
Catalog 2260
Prices $129.00
Sizes 5 mg
Function Type Antagonist
Cas Number 136054-22-3
Formula C49H63N13O6
Molecular Weight 930.12
Description Antagonist at the ghrelin receptor (GHS-R1a) (IC 50 = 0.9 μ M). Also weakly binds to melanocortin receptors (K i = 26-120 μ M). Centrally active in vivo .
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Product References

Characterization of the binding of MSH-B, HB-228, GHRP-6 and 153N-6 to the human - Characterization of the binding of MSH-B, HB-228, GHRP-6 and 153N-6 to the human

Schioth HB, Muceniece R, Wikberg JE. Neuropeptides. 1997 Dec;31(6):565-71.

Ghrelin acts on leptin-responsive neurones in the rat arcuate nucleus. - Ghrelin acts on leptin-responsive neurones in the rat arcuate nucleus.

Traebert M, Riediger T, Whitebread S, Scharrer E, Schmid HA. J Neuroendocrinol. 2002 Jul;14(7):580-6.

Role of ghrelin in the control of growth hormone secretion in prepubertal rats: - Role of ghrelin in the control of growth hormone secretion in prepubertal rats:

Pinilla L, Barreiro ML, Tena-Sempere M, Aguilar E. Neuroendocrinology. 2003 Feb;77(2):83-90.